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Антимикробные пептиды, нацеленные на липид II мембран бактерий: ключевой принцип действия
С. 60–60.
In book
Т. 2. , М.: Издательство "Перо", 2019.
Санина Н. А., Шилов Г. В., Ованесян Н. С. et al., Координационная химия 2023 Т. 49 № 9 С. 530–542
The synthesis and data on the physicochemical characteristics and biological activity of the new iron nitrosyl complex (Q+)2[Fe2(S2O3)2(NO)4]2– (I), where Q+ is protonated 2-ethyl-4-pyridinecarbothioamide (C8H11N2S), are presented. The structure and properties of the complex were studied by X-ray diffraction, elemental analysis, IR and Mössbauer spectroscopy, and amperometry. The complex showed antibacterial activity and efficiently inhibited ...
Added: September 14, 2025
Санина Н. А., Конюхова А. С., Корчагин Д. В. et al., Журнал неорганической химии 2023 Т. 68 № 9 С. 1165–1180
New neutral binuclear tetranitrosyl iron complexes of the composition [Fe2R2(NO)4] (R = 2,4-difluorothiophenyl(1) and 3,4-difluorothiophenyl(2)), donors of nitrogen oxide (NO), have been synthesized. The complexes were studied by Mossbauer, IR, and EPR spectroscopy, X-ray diffraction, and elemental analysis. The antibacterial activity and cytotoxicity in Vero cells of the complexes 1, 2 and the previously synthesized ...
Added: September 14, 2025
Козуб Г. И., Кондратьева Т. А., Шилов Г. В. et al., Известия Академии наук. Серия химическая 2023 Т. 72 № 3 С. 651–663
Three new binuclear tetranitrosyl iron complexes with m- and p-methoxybenzenethiolate and naphthalene-2-thiolate ligands have been synthesized. The crystals were characterized by X-ray diffraction, IR, Mossbauer spectroscopy, and elemental analysis. The NO-donating properties, cytotoxicity in tumor and non-cancerous cells, and antibacterial activity of the obtained complexes were studied. The toxicity of the complexes and the corresponding ...
Added: September 14, 2025
Forysenkova Anna A., Slukin P., Trofimchuk E. et al., Inorganic Materials: Applied Research 2023 Vol. 14 No. 2 P. 331–340
Powders of copper-, zinc-, manganese-substituted tricalcium phosphates (TCP) are synthesized; the composition and structure of the obtained compounds are studied. It is shown how copper, zinc, and manganese ions affect the phase composition and microstructure of substituted TCP powders. Composite materials based on a blend of polyvinylpyrrolidone with alginate (PVP:ALG) containing copper-, zinc-, and manganese-substituted ...
Added: August 13, 2025
Grechishnikova A., Слукин П. В., Трофимчук Е. С. et al., Перспективные материалы 2022 № 7 С. 35–48
Powders of copper, zinc, manganese-substituted tricalcium phosphates (TCP) were synthesized, the composition and structure of the obtained compounds were studied. It is shown how copper, zinc and manganese ions affect the phase composition and microstructure of powders substituted with TCP. Composite materials based on a blend of polyvinylpyrrolidone with alginate (PVP:ALG) containing copper, zinc, and ...
Added: August 12, 2025
Tsyklinskaya A. M., Polivanovskaia D. A., Grammatikova N. E. et al., Reactive and Functional Polymers 2024 Vol. 205 Article 106099
For the first time, a pronounced biocidal activity of modified polymers with a porphyrin content of 21.4 μM
(0.002 wt%) against Staphylococcus aureus was demonstrated. In order to develop new biocidal polymer coatings,
a study was carried out on diglycidyl ether of bisphenol A (DGEBA) and porphyrin-modified oligomeric diamine
systems. The study investigated the solubility of porphyrins in ...
Added: January 21, 2025
Русских С. В., Савлевич Е. Л., Васильева Т. П. et al., Якутский медицинский журнал 2024 № 3(87) С. 57–62
An algorithm for assessing the professional potential of an otorhinolaryngologist based on the identification of medical risk factors in the provision of medical care to patients with rhinosi-nusitis has been developed. otorhinolaryngologists from 32 subjects of the Russian Federation were screened and the treatment of patients with polyposis rhinosinusitis was analyzed. The proposed methodological approach ...
Added: October 8, 2024
Полянский А. А., Efremov R., Биологические мембраны 2024 Т. 41 № 4 С. 403–421
The paper overviews the results of computational studies of the molecular mechanisms underlying
the adaptation of model cell membranes taking place during their interaction with proteins and peptides. We
discuss changes in the structural and dynamic parameters of the water–lipid environment, the hydrophobic/
hydrophilic organization of the lipid bilayer surface (the so-called “mosaicity”), etc. Taken together,
these effects are ...
Added: September 19, 2024
Polyansky A. A., R. G. Efremov, Russian Journal of Bioorganic Chemistry 2024 Vol. 50 No. 4 P. 1202–1214
This study presents in a systematic manner the key modeling results corroborated by experimental
biophysical data and obtained by the authors during long-term research on bitopic (single-pass) membrane proteins
(BMPs), which are the crucial elements of cell signaling. The manuscript does not claim to be a comprehensive
review of the subject of interest, whereby the authors did not ...
Added: September 15, 2024
Gavira J. A., Rico-Jiménez M., Ortega A. et al., mBio 2023 Vol. 14 No. 1 Article e03363-22
Bacteria have evolved a sophisticated array of signal transduction systems that allow them to adapt their physiology and metabolism to changing environmental conditions. Typically, these systems recognize signals through dedicated ligand binding domains (LBDs) to ultimately trigger a diversity of physiological responses. Nonetheless, an increasing number of reports reveal that signal transduction receptors also bind ...
Added: January 27, 2024
Bershatsky Y., Kuznetsov A., Idiatullina A. et al., International Journal of Molecular Sciences 2023 Vol. 24 No. 4 Article 3906
Human InsR, IGF1R, and IRR receptor tyrosine kinases (RTK) of the insulin receptor
subfamily play an important role in signaling pathways for a wide range of physiological processes
and are directly associated with many pathologies, including neurodegenerative diseases. The
disulfide-linked dimeric structure of these receptors is unique among RTKs. Sharing high sequence
and structure homology, the receptors differ dramatically ...
Added: May 19, 2023
Abramov V., Abramova A., Bayazitov V. et al., Processes 2022 Vol. 10 No. 10 Article 2063
Although water contamination with drug residues is a threat to public health, there are currently barely any effective methods of purifying water from pharmaceutical substances. In this study, continuous-flow sonoplasma treatment was used for the complete degradation of tetracycline and ciprofloxacin in polluted municipal water. The addition of CeO2 nanoparticles as catalysts significantly increased the degradation ...
Added: October 23, 2022
Tharra P., Mikhaylov Andrey A., Švejkar J. et al., Angewandte Chemie - International Edition 2022 Vol. 61 No. 17 Article e202116520
Added: February 17, 2022
Lohan S., Mandal D., Choi W. et al., Journal of Medicinal Chemistry 2022 Vol. 65 No. 1 P. 665–687
We report the synthesis and antibacterial activities of a series of amphiphilic membrane-active peptides composed, in part, of various non-genetically coded hydrophobic amino acids. Lead cyclic peptides, 8C and 9C, showed broad-spectrum activity against drug-resistant Gram-positive (MIC=1.5-6.2 µg/mL) and Gram-negative (MIC=12.5-25 µg/mL) bacteria. Cytotoxicity study showed the predominant lethal action of the peptides against bacteria ...
Added: February 1, 2022
Ikonnikova V., Solyev P., Terekhov S. et al., ChemistrySelect 2021 Vol. 6 No. 42 P. 11775–11778
A short collective total synthesis of rearranged angucyclinones related to Elmenols A and B was achieved by ortho-lithiation/addition/transacetalisation sequence on the key step. Naphthalene and isocoumarine carbaldehydes required for synthesis were obtained in a straightforward manner by either of suitable methods: 1) palladium-catalyzed formylation, 2) halogen-lithium exchange, 3) decarboxylation of alpha-ketoacid. ...
Added: November 13, 2021
Omelchuk O., Malyshev V., Medvedev M. et al., Journal of Organic Chemistry 2021 Vol. 86 No. 12 P. 7975–7986
Oligomycin A is a potent antibiotic and antitumor agent. However, its applications are restricted by its high toxicity and low bioavailability. In this study, we obtained Oligomycin A Diels− Alder adducts with benzoquinone and N-benzylmaleimide and determined their absolute configurations by combining 1H and ROESY NMR data with molecular mechanics conformational analysis and quantum chemical ...
Added: September 6, 2021